Bioorganic and Medicinal Chemistry 2009
File List
- 9/sdarticle15.PDF 6.5 MB
- 14/Bora-Tatar_Molecular-modifications-on-carboxylic-acid-derivatives-as-potent-histone-deacetylase-inhibitors-Activity-and-docking-studies_2009.pdf 4.7 MB
- 2/sdarticle32.PDF 4.2 MB
- 13/Ahmed_Identification-of-novel-serotonin-2C-receptor-ligands-by-sequential-virtual-screening_2009.pdf 3.7 MB
- 16/Leung_Vancomycin-analogs-Seeking-improved-binding-of-d-Ala-d-Ala-and-d-Ala-d-Lac-peptides-by-side-chain-and-backbone-modifications_2009.pdf 3.7 MB
- 6/sdarticle20.PDF 3.7 MB
- 13/Zampieri_Antimycobacterial-activity-of-new-3,5-disubstituted-1,3,4-oxadiazol-2(3H)-one-derivatives.-Molecular-modeling-investigations_2009.pdf 3.6 MB
- 12/4160-4184.pdf 3.6 MB
- 15/Silvestri_Synthesis,-cannabinoid-receptor-affinity,-molecular-modeling-studies-and-in-vivo-pharmacological-evaluation-of-new-substituted-1-aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide.pdf 3.3 MB
- 8/sdarticle29.PDF 3.2 MB
- 13/Loizidou_Analysis-of-binding-parameters-of-HIV-1-integrase-inhibitors-Correlates-of-drug-inhibition-and-resistance_2009.pdf 3.2 MB
- 2/sdarticle48.PDF 3.1 MB
- 19/6851_6861.pdf 3.1 MB
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- 7/sdarticle19.PDF 2.9 MB
- 5/sdarticle23.PDF 2.8 MB
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- 18/Marchand_Synthesis-and-structure-activity-relationships-of-N-aryl(indol-3-yl)glyoxamides-as-antitumor-agents_2009.pdf 2.7 MB
- 19/7031_7041.pdf 2.5 MB
- 14/Ko_Molecular-recognition-in-the-P2Y14-receptor-Probing-the-structurally-permissive-terminal-sugar-moiety-of-uridine-5'-diphosphoglucose_2009.pdf 2.5 MB
- 6/sdarticle35.PDF 2.4 MB
- 13/Venkatraman_Discovery-of-novel-P3-sulfonamide-capped-inhibitors-of-HCV-NS3-protease.-Inhibitors-with-improved-cellular-potencies_2009.pdf 2.4 MB
- 10/sdarticle22.PDF 2.4 MB
- 20/7301-7312.pdf 2.4 MB
- 14/Michielan_Combining-selectivity-and-affinity-predictions-using-an-integrated-Support-Vector-Machine-(SVM)-approach-An-alternative-tool-to-discriminate-between-the-human-adenosine-A2A-and-A.pdf 2.3 MB
- 13/Barbayianni_2-Oxoamide-inhibitors-of-phospholipase-A2-activity-and-cellular-arachidonate-release-based-on-dipeptides-and-pseudodipeptides_2009.pdf 2.2 MB
- 1/2009_17/01/0165.pdf 2.2 MB
- 11/sdarticle10.PDF 2.2 MB
- 6/sdarticle43.PDF 2.2 MB
- 13/[first_author]_Graphical-contents-list_2009.pdf 2.2 MB
- 16/Abadi_Design,-synthesis-and-biological-evaluation-of-novel-pyridine-derivatives-as-anticancer-agents-and-phosphodiesterase-3-inhibitors_2009.pdf 2.1 MB
- 14/[first_author]_Graphical-contents-list_2009.pdf 2.1 MB
- 5/sdarticle22.PDF 2.1 MB
- 16/Prajapati_The-search-for-potent,-small-molecule-NNRTIs-A-review_2009.pdf 2.1 MB
- 14/Buttner_Synthesis-and-biological-evaluation-of-SANT-2-and-analogues-as-inhibitors-of-the-hedgehog-signaling-pathway_2009.pdf 2.0 MB
- 8/sdarticle16.PDF 2.0 MB
- 10/sdarticle23.PDF 2.0 MB
- 20/7290-7300.pdf 2.0 MB
- 6/sdarticle2.PDF 1.9 MB
- 13/Kirincich_Benzhydrylquinazolinediones-Novel-cytosolic-phospholipase-A2[alpha]-inhibitors-with-improved-physicochemical-properties_2009.pdf 1.9 MB
- 15/Ye_Discovery-of-novel-dual-functional-agent-as-PPAR[gamma]-agonist-and-11[beta]-HSD1-inhibitor-for-the-treatment-of-diabetes_2009.pdf 1.9 MB
- 9/sdarticle4.PDF 1.8 MB
- 4/sdarticle35.PDF 1.8 MB
- 14/Chen_Computational-selection-of-inhibitors-of-A[beta]-aggregation-and-neuronal-toxicity_2009.pdf 1.8 MB
- 5/sdarticle6.PDF 1.7 MB
- 11/sdarticle11.PDF 1.7 MB
- 12/4106-4126.pdf 1.7 MB
- 6/sdarticle53.PDF 1.7 MB
- 7/sdarticle11.PDF 1.7 MB
- 5/sdarticle35.PDF 1.7 MB
- 24/8206-8220.pdf 1.7 MB
- 20/7398-7404.pdf 1.7 MB
- 2/sdarticle11.PDF 1.7 MB
- 6/sdarticle39.PDF 1.7 MB
- 14/Haydar_SAR-and-biological-evaluation-of-SEN12333WAY-317538-Novel-alpha-7-nicotinic-acetylcholine-receptor-agonist_2009.pdf 1.7 MB
- 4/sdarticle24.PDF 1.7 MB
- 8/sdarticle26.PDF 1.7 MB
- 16/Seneci_Rational-design,-synthesis-and-characterization-of-potent,-non-peptidic-Smac-mimicsXIAP-inhibitors-as-proapoptotic-agents-for-cancer-therapy_2009.pdf 1.7 MB
- 19/6971_6982.pdf 1.6 MB
- 24/8221-8233.pdf 1.6 MB
- 13/Mou_Design,-synthesis-and-primary-activity-evaluation-of-l-arginine-derivatives-as-amino-peptidase-NCD13-inhibitors_2009.pdf 1.6 MB
- 16/Pan_A-comprehensive-study-of-Sansalvamide-A-derivatives-The-structure-activity-relationships-of-78-derivatives-in-two-pancreatic-cancer-cell-lines_2009.pdf 1.6 MB
- 20/7265-7274.pdf 1.6 MB
- 15/Lee_Antimicrobial-natural-products-as-[beta]-ketoacyl-acyl-carrier-protein-synthase-III-inhibitors_2009.pdf 1.6 MB
- 18/Tasler_Substituted-2-arylbenzothiazoles-as-kinase-inhibitors-Hit-to-lead-optimization_2009.pdf 1.6 MB
- 8/sdarticle24.PDF 1.5 MB
- 4/sdarticle2.PDF 1.5 MB
- 16/[first_author]_Graphical-contents-list_2009.pdf 1.5 MB
- 15/[first_author]_Graphical-contents-list_2009.pdf 1.5 MB
- 5/sdarticle24.PDF 1.5 MB
- 14/Marcelo_Synthesis-of-novel-purine-nucleosides-towards-a-selective-inhibition-of-human-butyrylcholinesterase_2009.pdf 1.5 MB
- 1/2009_17/01/0401.pdf 1.5 MB
- 5/sdarticle2.PDF 1.5 MB
- 2/sdarticle24.PDF 1.5 MB
- 2/sdarticle18.PDF 1.5 MB
- 12/4035-4046.pdf 1.5 MB
- 18/Kim_A-new-structural-class-of-S-adenosylhomocysteine-hydrolase-inhibitors_2009.pdf 1.5 MB
- 22/7795-7801.pdf 1.5 MB
- 18/Asada_Discovery-of-a-series-of-acrylic-acids-and-their-derivatives-as-chemical-leads-for-selective-EP3-receptor-antagonists_2009.pdf 1.5 MB
- 7/sdarticle32.PDF 1.4 MB
- 15/Joeng_ssDNA-aptamers-that-recognize-diclofenac-and-2-anilinophenylacetic-acid_2009.pdf 1.4 MB
- 19/7042_7051.pdf 1.4 MB
- 9/sdarticle19.PDF 1.4 MB
- 21/7465_7476.pdf 1.4 MB
- 4/sdarticle25.PDF 1.4 MB
- 9/sdarticle3.PDF 1.4 MB
- 4/sdarticle15.PDF 1.4 MB
- 9/sdarticle18.PDF 1.4 MB
- 23/7933.pdf 1.4 MB
- 15/Yongye_Identification,-structure-activity-relationships-and-molecular-modeling-of-potent-triamine-and-piperazine-opioid-ligands_2009.pdf 1.4 MB
- 19/6959_6970.pdf 1.4 MB
- 3/sdarticle2.PDF 1.4 MB
- 17/[first_author]_Graphical-contents-list_2009.pdf 1.4 MB
- 1/2009_17/01/0149.pdf 1.4 MB
- 15/Trayner_Synthesis-and-characterization-of-6-deoxy-6-fluoro-d-fructose-as-a-potential-compound-for-imaging-breast-cancer-with-PET_2009.pdf 1.4 MB
- 10/sdarticle13.PDF 1.3 MB
- 20/7075-7084.pdf 1.3 MB
- 10/sdarticle14.PDF 1.3 MB
- 7/sdarticle2.PDF 1.3 MB
- 16/Novak_Free-and-bound-state-structures-of-6-O-methyl-homoerythromycins-and-epitope-mapping-of-their-interactions-with-ribosomes_2009.pdf 1.3 MB
- 20/7368-7380.pdf 1.3 MB
- 17/Mosley_Synthesis,-structural-activity-relationships,-and-biological-evaluation-of-novel-amide-based-allosteric-binding-site-antagonists-in-NR1ANR2B-N-methyl-d-aspartate-receptors_2009.pdf 1.3 MB
- 7/sdarticle5.PDF 1.3 MB
- 11/sdarticle27.PDF 1.3 MB
- 16/Gleeson_ADMET-rules-of-thumb-II-A-comparison-of-the-effects-of-common-substituents-on-a-range-of-ADMET-parameters_2009.pdf 1.3 MB
- 22/7732-7742.pdf 1.3 MB
- 12/4241-4256.pdf 1.3 MB
- 19/6926_6936.pdf 1.3 MB
- 18/[first_author]_Graphical-contents-list_2009.pdf 1.3 MB
- 1/2009_17/01/0176.pdf 1.3 MB
- 16/Gemma_Development-of-antitubercular-compounds-based-on-a-4-quinolylhydrazone-scaffold.-Further-structure-activity-relationship-studies_2009.pdf 1.3 MB
- 9/sdarticle30.PDF 1.3 MB
- 14/Zhao_Diketoacid-genre-HIV-1-integrase-inhibitors-containing-enantiomeric-arylamide-functionality_2009.pdf 1.2 MB
- 14/Trapella_Structure-activity-studies-on-the-nociceptinorphanin-FQ-receptor-antagonist-1-benzyl-N-{3-[spiroisobenzofuran-1(3H),4'-piperidin-1-yl]propyl}-pyrrolidine-2-carboxamide_2009.pdf 1.2 MB
- 8/sdarticle3.PDF 1.2 MB
- 2/sdarticle2.PDF 1.2 MB
- 20/7174-7185.pdf 1.2 MB
- 19/6787_6795.pdf 1.2 MB
- 13/Chen_Synthetic-resveratrol-aliphatic-acid-inhibits-TLR2-mediated-apoptosis-and-an-involvement-of-AktGSK3[beta]-pathway_2009.pdf 1.2 MB
- 10/sdarticle2.PDF 1.2 MB
- 21/7457_7464.pdf 1.2 MB
- 16/Khanfar_The-marine-natural-derived-inhibitors-of-glycogen-synthase-kinase-3[beta]-phenylmethylene-hydantoins-In-vitro-and-in-vivo-activities-and-pharmacophore-modeling_2009.pdf 1.2 MB
- 14/Sakamoto_Novel-orally-active-NPY-Y5-receptor-antagonists-Synthesis-and-structure-activity-relationship-of-spiroindoline-class-compounds_2009.pdf 1.2 MB
- 15/Ngoupayo_Antimicrobial-and-immunomodulatory-properties-of-prenylated-xanthones-from-twigs-of-Garcinia-staudtii_2009.pdf 1.2 MB
- 8/sdarticle2.PDF 1.2 MB
- 7/sdarticle36.PDF 1.2 MB
- 9/sdarticle20.PDF 1.2 MB
- 19/6983_6992.pdf 1.2 MB
- 13/Aiello_Discovery,-characterization-and-comparison-of-inhibitors-of-Bacillus-anthracis-and-Staphylococcus-aureus-replicative-DNA-helicases_2009.pdf 1.2 MB
- 16/Ando_Discovery-of-pyridone-containing-imidazolines-as-potent-and-selective-inhibitors-of-neuropeptide-Y-Y5-receptor_2009.pdf 1.2 MB
- 6/sdarticle4.PDF 1.2 MB
- 23/7841.pdf 1.2 MB
- 13/Toth_Synthesis-and-structure-activity-relationships-of-C-glycosylated-oxadiazoles-as-inhibitors-of-glycogen-phosphorylase_2009.pdf 1.2 MB
- 22/7831-7840.pdf 1.2 MB
- 17/Gouda_Molecular-modeling-of-human-acidic-mammalian-chitinase-in-complex-with-the-natural-product-cyclopentapeptide-chitinase-inhibitor-argifin_2009.pdf 1.2 MB
- 10/sdarticle10.PDF 1.2 MB
- 6/sdarticle49.PDF 1.2 MB
- 16/Huang_Synthesis,-DNA-intercalation-and-3D-QSAR-analysis-of-cis-2,4,5-trisubstituted-1,3-dithiolanes-as-a-novel-class-of-antitumor-agents_2009.pdf 1.1 MB
- 23/7924.pdf 1.1 MB
- 19/7021_7030.pdf 1.1 MB
- 13/Kuder_Synthesis-and-biological-activity-of-a-fluorescent-schweinfurthin-analogue_2009.pdf 1.1 MB
- 1/2009_17/01/0085.pdf 1.1 MB
- 11/sdarticle2.PDF 1.1 MB
- 18/Ngen_Evaluation-of-delocalized-lipophilic-cationic-dyes-as-delivery-vehicles-for-photosensitizers-to-mitochondria_2009.pdf 1.1 MB
- 12/4071-4084.pdf 1.1 MB
- 5/sdarticle3.PDF 1.1 MB
- 18/Gillespie_Antagonists-of-the-human-A2A-receptor.-Part-6-Further-optimization-of-pyrimidine-4-carboxamides_2009.pdf 1.1 MB
- 19/6898_6907.pdf 1.1 MB
- 5/sdarticle31.PDF 1.1 MB
- 18/Shah_Synthesis,-structure-affinity-relationships,-and-modeling-of-AMDA-analogs-at-5-HT2A-and-H1-receptors-Structural-factors-contributing-to-selectivity_2009.pdf 1.1 MB
- 12/4197-4205.pdf 1.1 MB
- 16/Hasegawa_A-highly-sensitive-probe-detecting-low-pH-area-of-HeLa-cells-based-on-rhodamine-B-modified-[beta]-cyclodextrins_2009.pdf 1.1 MB
- 13/Magesh_Human-sialidase-inhibitors-Design,-synthesis,-and-biological-evaluation-of-4-acetamido-5-acylamido-2-fluoro-benzoic-acids_2009.pdf 1.1 MB
- 5/sdarticle34.PDF 1.1 MB
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- 19/6914_6925.pdf 1.0 MB
- 1/2009_17/01/0326.pdf 1.0 MB
- 15/Noeske_Synergism-of-virtual-screening-and-medicinal-chemistry-Identification-and-optimization-of-allosteric-antagonists-of-metabotropic-glutamate-receptor-1_2009.pdf 1.0 MB
- 11/sdarticle23.PDF 1.0 MB
- 15/Oka_Syntheses-and-biological-evaluations-of-carbosilane-dendrimers-uniformly-functionalized-with-sialyl-[alpha](2--3)-lactose-moieties-as-inhibitors-for-human-influenza-viruses_2009.pdf 1.0 MB
- 1/2009_17/01/0013.pdf 1.0 MB
- 7/sdarticle28.PDF 1.0 MB
- 16/Deb_Synthesis-and-characterizations-of-novel-quinoline-derivatives-having-mixed-ligand-activities-at-the-[kappa]-and-[mu]-receptors-Potential-therapeutic-efficacy-against-morphine-dependen.pdf 1020.8 KB
- 22/7769-7774.pdf 1016.3 KB
- 9/sdarticle5.PDF 998.8 KB
- 16/Harada_Evaluation-of-hydrogen-bonds-of-ecdysteroids-in-the-ligand-receptor-interactions-using-a-protein-modeling-system_2009.pdf 998.7 KB
- 21/7405_7411.pdf 994.4 KB
- 8/sdarticle6.PDF 994.3 KB
- 21/7412_7417.pdf 994.3 KB
- 20/7324-7336.pdf 993.9 KB
- 15/Sasaki_Synthesis-and-evaluation-of-a-novel-2-azabicyclo[2.2.2]octane-class-of-long-chain-fatty-acid-elongase-6-(ELOVL6)-inhibitors_2009.pdf 992.8 KB
- 21/7593_7605.pdf 990.3 KB
- 21/7441_7448.pdf 989.6 KB
- 20/7197-7208.pdf 986.4 KB
- 6/sdarticle29.PDF 983.4 KB
- 11/sdarticle34.PDF 965.6 KB
- 8/sdarticle5.PDF 963.6 KB
- 15/Sakamoto_Systematic-syntheses-of-influenza-neuraminidase-inhibitors-A-series-of-carbosilane-dendrimers-uniformly-functionalized-with-thioglycoside-type-sialic-acid-moieties_2009.pdf 961.9 KB
- 9/sdarticle21.PDF 958.4 KB
- 5/sdarticle37.PDF 948.0 KB
- 7/sdarticle33.PDF 940.1 KB
- 20/7100-7107.pdf 939.4 KB
- 15/Itoh_Inhibitory-effects-of-flavonoids-isolated-from-Fragaria-ananassa-Duch-on-IgE-mediated-degranulation-in-rat-basophilic-leukemia-RBL-2H3_2009.pdf 939.2 KB
- 11/sdarticle16.PDF 937.4 KB
- 5/sdarticle12.PDF 932.6 KB
- 9/sdarticle25.PDF 930.9 KB
- 17/Shomin_Staurosporine-tethered-peptide-ligands-that-target-cAMP-dependent-protein-kinase-(PKA)-Optimization-and-selectivity-profiling_2009.pdf 929.9 KB
- 22/7658-7669.pdf 926.2 KB
- 19/6952_6958.pdf 918.8 KB
- 21/7523_7530.pdf 918.8 KB
- 14/Daines_Mannosylated-saponins-based-on-oleanolic-and-glycyrrhizic-acids.-Towards-synthetic-colloidal-antigen-delivery-systems_2009.pdf 917.1 KB
- 1/2009_17/01/0074.pdf 915.8 KB
- 23/8060.pdf 914.0 KB
- 6/sdarticle52.PDF 913.6 KB
- 14/Zhu_Quantitative-high-throughput-screening-identifies-inhibitors-of-anthrax-induced-cell-death_2009.pdf 912.5 KB
- 7/sdarticle22.PDF 911.0 KB
- 22/Graphical contents list.pdf 908.5 KB
- 14/El-Shafei_Synthesis,-antitumor-evaluation,-molecular-modeling-and-quantitative-structure-activity-relationship-(QSAR)-of-some-novel-arylazopyrazolodiazine-and-triazine-analogs_2009.pdf 904.1 KB
- 17/Santos_Novel-semisynthetic-derivatives-of-betulin-and-betulinic-acid-with-cytotoxic-activity_2009.pdf 903.1 KB
- 3/sdarticle10.PDF 902.5 KB
- 17/van-der-Knaap_Synthesis-and-biological-evaluation-of-asymmetric-gramicidin-S-analogues-containing-modified-d-phenylalanine-residues_2009.pdf 901.0 KB
- 18/Riveiro_Toward-establishing-structure-activity-relationships-for-oxygenated-coumarins-as-differentiation-inducers-of-promonocytic-leukemic-cells_2009.pdf 895.2 KB
- 2/sdarticle33.PDF 890.4 KB
- 15/Kakadiya_Potent-antitumor-bifunctional-DNA-alkylating-agents,-synthesis-and-biological-activities-of-3a-aza-cyclopenta[a]indenes_2009.pdf 890.2 KB
- 6/sdarticle51.PDF 888.4 KB
- 12/4206-4215.pdf 884.8 KB
- 4/sdarticle29.PDF 884.8 KB
- 7/sdarticle14.PDF 884.5 KB
- 6/sdarticle22.PDF 879.3 KB
- 23/7978.pdf 878.0 KB
- 3/sdarticle6.PDF 868.9 KB
- 8/sdarticle18.PDF 867.6 KB
- 16/Jhansi-Lakshmi_Design,-synthesis,-and-discovery-of-novel-non-peptide-inhibitor-of-Caspase-3-using-ligand-based-and-structure-based-virtual-screening-approach_2009.pdf 866.9 KB
- 2/sdarticle6.PDF 865.6 KB
- 6/sdarticle25.PDF 861.2 KB
- 16/Singh_Reactions-of-hydroxyl-radical-with-bergenin,-a-natural-poly-phenol-studied-by-pulse-radiolysis_2009.pdf 858.3 KB
- 23/7964.pdf 856.8 KB
- 13/Zheng_QSAR-study-on-maximal-inhibition-(Imax)-of-quaternary-ammonium-antagonists-for-S-(-)-nicotine-evoked-dopamine-release-from-dopaminergic-nerve-terminals-in-rat-striatum_2009.pdf 851.3 KB
- 16/Gigante_SAR-studies-on-azasterols-as-potential-anti-trypanosomal-and-anti-leishmanial-agents_2009.pdf 850.9 KB
- 13/Alvarez_Retinoid-receptor-subtype-selective-modulators-through-synthetic-modifications-of-RAR[gamma]-agonists_2009.pdf 848.2 KB
- 13/Tonelli_Antiviral-and-cytotoxic-activities-of-aminoarylazo-compounds-and-aryltriazene-derivatives_2009.pdf 847.5 KB
- 3/sdarticle19.PDF 844.8 KB
- 7/sdarticle24.PDF 844.6 KB
- 14/Liu_Characterization-and-synthetic-application-of-a-novel-[beta]1,3-galactosyltransferase-from-Escherichia-coli-O55H7_2009.pdf 844.4 KB
- 8/sdarticle15.PDF 843.6 KB
- 3/sdarticle22.PDF 837.0 KB
- 2/sdarticle46.PDF 835.8 KB
- 9/sdarticle7.PDF 833.4 KB
- 13/Gao_Synthesis-and-biological-evaluation-of-novel-carbon-11-labeled-pyridyl-ethers-candidate-ligands-for-in-vivo-imaging-of-[alpha]4[beta]2-nicotinic-acetylcholine-receptors-([alpha]4[beta].pdf 832.1 KB
- 16/Cox_Characterization-and-DNA-interaction-studies-of-1,1-dicyano-2,2-ethylene-dithiolate-Ni(II)-mixed-ligand-complexes-with-2-amino-5-methyl-thiazole,-2-amino-2-thiazoline-and-imidazole.-Cr.pdf 831.2 KB
- 17/Koufaki_Design-and-synthesis-of-novel-neuroprotective-1,2-dithiolanechroman-hybrids_2009.pdf 828.5 KB
- 4/sdarticle36.PDF 826.2 KB
- 7/sdarticle12.PDF 825.0 KB
- 16/Orrling_[alpha]-Substituted-norstatines-as-the-transition-state-mimic-in-inhibitors-of-multiple-digestive-vacuole-malaria-aspartic-proteases_2009.pdf 819.0 KB
- 10/sdarticle27.PDF 818.7 KB
- 21/7548_7561.pdf 816.0 KB
- 4/sdarticle13.PDF 815.7 KB
- 5/sdarticle25.PDF 815.4 KB
- 4/sdarticle43.PDF 812.9 KB
- 10/sdarticle24.PDF 810.8 KB
- 2/sdarticle3.PDF 808.9 KB
- 17/Yang_Artemetherhydroxypropyl-[beta]-cyclodextrin-host-guest-system-Characterization,-phase-solubility-and-inclusion-mode_2009.pdf 807.8 KB
- 19/6841_6850.pdf 804.6 KB
- 15/Spathelf_Anti-listerial-activity-and-structure-activity-relationships-of-the-six-major-tyrocidines,-cyclic-decapeptides-from-Bacillus-aneurinolyticus_2009.pdf 800.5 KB
- 22/7711-7722.pdf 799.8 KB
- 4/sdarticle11.PDF 798.2 KB
- 20/7085-7092.pdf 797.8 KB
- 18/Gokhan-Kelekci_Synthesis-and-molecular-modeling-of-some-novel-hexahydroindazole-derivatives-as-potent-monoamine-oxidase-inhibitors_2009.pdf 796.2 KB
- 22/7743-7748.pdf 791.0 KB
- 14/Bertucci_Carbonic-anhydrase-inhibitors.-Inhibition-studies-of-a-coral-secretory-isoform-by-sulfonamides_2009.pdf 790.7 KB
- 24/8186-8196.pdf 784.8 KB
- 6/sdarticle46.PDF 782.6 KB
- 13/Henry_A-versatile-photoactivatable-probe-designed-to-label-the-diphosphate-binding-site-of-farnesyl-diphosphate-utilizing-enzymes_2009.pdf 781.8 KB
- 15/Patel_Interaction-of-drug-based-binuclear-mixed-ligand-complexes-with-DNA_2009.pdf 779.6 KB
- 12/4013-4018.pdf 767.2 KB
- 18/Todoroki_Abscinazole-F1,-a-conformationally-restricted-analogue-of-the-plant-growth-retardant-uniconazole-and-an-inhibitor-of-ABA-8'-hydroxylase-CYP707A-with-no-growth-retardant-effect_200.pdf 766.6 KB
- 21/7615_7621.pdf 766.2 KB
- 23/8020.pdf 761.7 KB
- 19/7064_7072.pdf 761.5 KB
- 1/2009_17/01/0001.pdf 761.3 KB
- 5/sdarticle16.PDF 758.5 KB
- 16/Sato_Synthesis,-biological-evaluation,-and-metabolic-stability-of-acrylamide-derivatives-as-novel-CCR3-antagonists_2009.pdf 753.2 KB
- 14/Maie_Fluorescence-quenching-properties-of-multiple-pyrene-modified-RNAs_2009.pdf 748.8 KB
- 14/Debnath_Nucleoside-amino-acid-conjugates-An-alternative-route-to-the-design-of-ribonuclease-A-inhibitors_2009.pdf 748.1 KB
- 24/8174-8185.pdf 747.5 KB
- 9/sdarticle29.PDF 742.9 KB
- 4/sdarticle8.PDF 740.8 KB
- 22/7755-7768.pdf 739.0 KB
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- 14/Hadjipavlou-Litina_2D-QSAR-and-3D-QSARCoMFA-analyses-of-the-N-terminal-substituted-anthranilic-acid-based-CCK1-receptor-antagonists-`Hic-Rhodus,-hic-saltus'_2009.pdf 731.4 KB
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- 15/Corbel_Identification-of-potential-cellular-targets-of-aloisine-A-by-affinity-chromatography_2009.pdf 723.6 KB
- 13/Ohkubo_Efficient-solid-phase-synthesis-of-oligodeoxynucleotides-having-a-5'-terminal-2,2,7-trimethylguanosine-pyrophosphate-linkage_2009.pdf 722.6 KB
- 12/4085-4095.pdf 719.4 KB
- 14/Minond_Inhibitors-of-VIM-2-by-screening-pharmacologically-active-and-click-chemistry-compound-libraries_2009.pdf 715.6 KB
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- 15/Mourer_p-Guanidinoethyl-calixarene-and-parent-phenol-derivatives-exhibiting-antibacterial-activities.-Synthesis-and-biological-evaluation_2009.pdf 713.6 KB
- 2/sdarticle50.PDF 712.7 KB
- 17/Zhao_N-[2-Chloro-9H-purin-6-yl]-N-cyclopropylglycylamino-acids-and-derivatives-Synthesis,-evaluation-as-a-class-of-novel-analgesics,-and-3D-QSAR-analysis_2009.pdf 710.9 KB
- 17/Hockova_Synthesis-of-branched-9-[2-(2-phosphonoethoxy)ethyl]purines-as-a-new-class-of-acyclic-nucleoside-phosphonates-which-inhibit-Plasmodium-falciparum-hypoxanthine-guanine-xanthine-phos.pdf 710.3 KB
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- 17/Li_Synthesis-of-C(7)-modified-chrysin-derivatives-designing-to-inhibit-[beta]-ketoacyl-acyl-carrier-protein-synthase-III-(FabH)-as-antibiotics_2009.pdf 680.3 KB
- 14/Motoshima_Separation-of-[alpha]-glucosidase-inhibitory-and-liver-X-receptor-antagonistic-activities-of-phenethylphenyl-phthalimide-analogs-and-generation-of-LXR[alpha]-selective-antagonist.pdf 679.7 KB
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- 1/2009_17/01/0284.pdf 675.9 KB
- 15/Azema_7-((4-Substituted)piperazin-1-yl)-derivatives-of-ciprofloxacin-Synthesis-and-in-vitro-biological-evaluation-as-potential-antitumor-agents_2009.pdf 675.7 KB
- 14/Berenguer_Tetrahydroisoquinolines-as-dopaminergic-ligands-1-Butyl-7-chloro-6-hydroxy-tetrahydroisoquinoline,-a-new-compound-with-antidepressant-like-activity-in-mice_2009.pdf 673.8 KB
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- 13/Ronco_Synthesis-and-structure-activity-relationship-of-Huprine-derivatives-as-human-acetylcholinesterase-inhibitors_2009.pdf 664.4 KB
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- 14/Ananda-Kumar_Anti-tumor-and-anti-angiogenic-activity-of-novel-hydantoin-derivatives-Inhibition-of-VEGF-secretion-in-liver-metastatic-osteosarcoma-cells_2009.pdf 662.3 KB
- 21/7572_7584.pdf 661.1 KB
- 10/sdarticle29.PDF 660.4 KB
- 13/Glavas-Obrovac_Minor-structural-differences-of-monomethine-cyanine-derivatives-yield-strong-variation-in-their-interactions-with-DNA,-RNA-as-well-as-on-their-in-vitro-antiproliferative-act.pdf 658.2 KB
- 15/Simunovic_Urea-and-carbamate-derivatives-of-primaquine-Synthesis,-cytostatic-and-antioxidant-activities_2009.pdf 656.0 KB
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- 16/Misra_Immobilization-of-self-quenched-DNA-hairpin-probe-with-a-heterobifunctional-reagent-on-a-glass-surface-for-sensitive-detection-of-oligonucleotides_2009.pdf 649.4 KB
- 2/sdarticle39.PDF 648.8 KB
- 13/Yu_Phage-display-screening-against-a-set-of-targets-to-establish-peptide-based-sugar-mimetics-and-molecular-docking-to-predict-binding-site_2009.pdf 648.6 KB
- 19/7056_7063.pdf 647.2 KB
- 1/2009_17/01/0042.pdf 646.0 KB
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- 15/Li_Design-and-synthesis-of-acetamido-tri--and-tetra-hydroxyazepanes-Potent-and-selective-[beta]-N-acetylhexosaminidase-inhibitors_2009.pdf 640.8 KB
- 14/Kranz_Identification-of-PDE4B-Over-4D-subtype-selective-inhibitors-revealing-an-unprecedented-binding-mode_2009.pdf 640.8 KB
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- 17/Alvarez_Isocombretastatins-A-1,1-Diarylethenes-as-potent-inhibitors-of-tubulin-polymerization-and-cytotoxic-compounds_2009.pdf 636.4 KB
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- 17/Tuin_Structural-and-biological-evaluation-of-some-loloatin-C-analogues_2009.pdf 635.7 KB
- 13/Erez_Enhanced-cytotoxicity-of-a-polymer-drug-conjugate-with-triple-payload-of-paclitaxel_2009.pdf 633.2 KB
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- 15/Su_Effects-of-structural-analogues-of-the-substrate-and-allosteric-regulator-of-the-human-mitochondrial-NAD(P)+-dependent-malic-enzyme_2009.pdf 625.8 KB
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- 14/Oishi_Design-and-synthesis-of-membrane-fusion-inhibitors-against-the-feline-immunodeficiency-virus_2009.pdf 619.3 KB
- 17/Peng_Novel-delta-opioid-receptor-agonists-exhibit-differential-stimulation-of-signaling-pathways_2009.pdf 616.9 KB
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- 16/Fujii_Aerobic-oxidation-of-indolomorphinan-without-the-4,5-epoxy-bridge-and-subsequent-rearrangement-of-the-oxidation-product-to-spiroindolinonyl-C-normorphinan-derivative_2009.pdf 613.4 KB
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- 18/Ikeuchi_A-critical-electrostatic-interaction-mediates-inhibitor-recognition-by-human-asparagine-synthetase_2009.pdf 610.3 KB
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- 16/Aubry_Fascaplysin-inspired-diindolyls-as-selective-inhibitors-of-CDK4cyclin-D1_2009.pdf 608.2 KB
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- 16/Hazai_A-comprehensive-study-on-the-5-hydroxytryptamine3A-receptor-binding-of-agonists-serotonin-and-m-chlorophenylbiguanidine_2009.pdf 605.5 KB
- 13/Moran_Synthesis,-structural-characterisation-and-biological-evaluation-of-fluorinated-analogues-of-resveratrol_2009.pdf 603.5 KB
- 15/Fuchigami_Development-of-N-[11C]methylamino-4-hydroxy-2(1H)-quinolone-derivatives-as-PET-radioligands-for-the-glycine-binding-site-of-NMDA-receptors_2009.pdf 601.4 KB
- 14/Sun_Synthesis-and-multidrug-resistance-reversal-activity-of-dihydroptychantol-A-and-its-novel-derivatives_2009.pdf 600.6 KB
- 18/Debnath_Inhibition-of-ribonuclease-A-by-nucleoside-dibasic-acid-conjugates_2009.pdf 599.8 KB
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- 14/Ebalunode_Structure-based-shape-pharmacophore-modeling-for-the-discovery-of-novel-anesthetic-compounds_2009.pdf 576.9 KB
- 4/sdarticle18.PDF 576.7 KB
- 16/Abeydeera_Synthesis-and-characterization-of-modified-nucleotides-in-the-970-hairpin-loop-of-Escherichia-coli-16S-ribosomal-RNA_2009.pdf 576.2 KB
- 3/sdarticle5.PDF 574.1 KB
- 18/Maia_Synthesis-and-analgesic-profile-of-conformationally-constrained-N-acylhydrazone-analogues-Discovery-of-novel-N-arylideneamino-quinazolin-4(3H)-one-compounds-derived-from-natural-safro.pdf 573.9 KB
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- 14/Zhang_Bioactive-conformation-analysis-of-cyclic-imides-as-protoporphyrinogen-oxidase-inhibitor-by-combining-DFT-calculations,-QSAR-and-molecular-dynamic-simulations_2009.pdf 561.9 KB
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- 16/Foss-Jr._Synthesis-and-biological-evaluation-of-sphingosine-kinase-substrates-as-sphingosine-1-phosphate-receptor-prodrugs_2009.pdf 555.2 KB
- 8/sdarticle7.PDF 554.6 KB
- 17/Wang_Preparation-of-C-23-esterified-silybin-derivatives-and-evaluation-of-their-lipid-peroxidation-inhibitory-and-DNA-protective-properties_2009.pdf 552.8 KB
- 20/7113-7125.pdf 551.8 KB
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- 13/Ye_Synthesis-and-biological-evaluation-of-novel-4-azaindolyl-indolyl-maleimides-as-glycogen-synthase-kinase-3[beta]-(GSK-3[beta])-inhibitors_2009.pdf 541.7 KB
- 14/Nielsen_An-extended-study-of-dimeric-phenyl-tropanes_2009.pdf 541.3 KB
- 13/Ye_Synthesis-and-evaluation-of-novel-7-azaindazolyl-indolyl-maleimide-derivatives-as-antitumor-agents-and-protein-kinase-C-inhibitors_2009.pdf 541.1 KB
- 23/8102.pdf 540.3 KB
- 13/Perez-Cruz_Molecular-encapsulation-of-5-nitroindazole-derivatives-in-2,6-dimethyl-[beta]-cyclodextrin-Electrochemical-and-spectroscopic-studies_2009.pdf 538.9 KB
- 24/8161-8167.pdf 538.9 KB
- 5/sdarticle15.PDF 538.6 KB
- 17/Wada_Anti-tumor-initiating-effects-of-phenolic-compounds-isolated-from-the-bark-of-Picea-jezoensis-var.-jezoensis_2009.pdf 538.4 KB
- 7/sdarticle3.PDF 538.3 KB
- 17/Tashiro_RCAI-37,-56,-59,-60,-92,-101,-and-102,-cyclitol-and-carbasugar-analogs-of-KRN7000-Their-synthesis-and-bioactivity-for-mouse-lymphocytes-to-produce-Th1-biased-cytokines_2009.pdf 538.1 KB
- 10/sdarticle25.PDF 538.0 KB
- 13/Shao_Synthesis-and-DNA-cleavage-activity-of-2-hydrazinyl-1,4,5,6-tetrahydropyrimidine-containing-hydroxy-group_2009.pdf 537.6 KB
- 5/sdarticle13.PDF 537.5 KB
- 13/Jiao_Lathyrane-diterpenes-from-Euphorbia-lathyris-as-modulators-of-multidrug-resistance-and-their-crystal-structures_2009.pdf 535.0 KB
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- 14/Kumar_Design-and-synthesis-of-3,5-diarylisoxazole-derivatives-as-novel-class-of-anti-hyperglycemic-and-lipid-lowering-agents_2009.pdf 525.2 KB
- 5/sdarticle9.PDF 524.0 KB
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- 1/2009_17/01/0344.pdf 518.6 KB
- 14/Kontijevskis_Proteochemometrics-mapping-of-the-interaction-space-for-retroviral-proteases-and-their-substrates_2009.pdf 518.4 KB
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- 15/Sethi_Polymer-supported-synthesis-of-aminooxyalkylated-oligonucleotides,-and-some-applications-in-the-fabrication-of-microarrays_2009.pdf 511.4 KB
- 18/dos-Santos-Filho_Design,-synthesis-and-cruzain-docking-of-3-(4-substituted-aryl)-1,2,4-oxadiazole-N-acylhydrazones-as-anti-Trypanosoma-cruzi-agents_2009.pdf 509.9 KB
- 13/De-Wael_In-vitro-and-in-vivo-studies-of-6,8-(diaryl)imidazo[1,2-a]pyrazin-3(7H)-ones-as-new-antioxidants_2009.pdf 507.7 KB
- 17/Szymanska_3-Substituted-phenylalanines-as-selective-AMPA--and-kainate-receptor-ligands_2009.pdf 506.9 KB
- 24/8241-8246.pdf 506.7 KB
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- 13/Karis_Glycogen-phosphorylase-inhibitory-effects-of-2-oxo-1,2-dihydropyridin-3-yl-amide-derivatives_2009.pdf 505.2 KB
- 8/sdarticle19.PDF 504.0 KB
- 13/Reux_Synthesis-of-quinolinyl-and-isoquinolinyl-phenyl-ketones-as-novel-agonists-for-the-cannabinoid-CB2-receptor_2009.pdf 503.8 KB
- 13/Shim_Inhibitory-effects-of-phloroglucinol-derivatives-isolated-from-Ecklonia-stolonifera-on-Fc[epsilon]RI-expression_2009.pdf 503.6 KB
- 11/sdarticle14.PDF 502.0 KB
- 17/Caruso_Inhibitory-effect-of-[beta]-diketones-and-their-metal-complexes-on-TNF-[alpha]-induced-expression-of-ICAM-1-on-human-endothelial-cells_2009.pdf 501.9 KB
- 13/Upadhayaya_Design,-synthesis-and-biological-evaluation-of-novel-triazole,-urea-and-thiourea-derivatives-of-quinoline-against-Mycobacterium-tuberculosis_2009.pdf 501.3 KB
- 2/sdarticle30.PDF 500.8 KB
- 17/Claramunt_Fluorinated-indazoles-as-novel-selective-inhibitors-of-nitric-oxide-synthase-(NOS)-Synthesis-and-biological-evaluation_2009.pdf 500.5 KB
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- 20/7209-7217.pdf 499.4 KB
- 14/Mora-Pale_Inhibition-of-human-vascular-NADPH-oxidase-by-apocynin-derived-oligophenols_2009.pdf 497.2 KB
- 6/sdarticle42.PDF 496.5 KB
- 15/Maruyama_Discovery-of-novel-thiourea-derivatives-as-potent-and-selective-[beta]3-adrenergic-receptor-agonists_2009.pdf 495.6 KB
- 3/sdarticle51.PDF 495.3 KB
- 13/Crepaldi_6-Amino-2-mercapto-3H-pyrimidin-4-one-derivatives-as-new-candidates-for-the-antagonism-at-the-P2Y12-receptors_2009.pdf 494.4 KB
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- 16/Zhan_Novel-1,2,3-thiadiazole-derivatives-as-HIV-1-NNRTIs-with-improved-potency-Synthesis-and-preliminary-SAR-studies_2009.pdf 491.5 KB
- 11/sdarticle6.PDF 491.1 KB
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- 16/Shoji_Novel-indoline-based-acyl-CoA-cholesterol-acyltransferase-inhibitor-Effects-of-introducing-a-methanesulfonamide-group-on-physicochemical-properties-and-biological-activities_2009.pdf 489.4 KB
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- 13/Willemann_Synthesis-and-cytotoxic-activity-of-5,6-heteroaromatically-annulated-pyridine-2,4-diamines_2009.pdf 484.8 KB
- 18/Micale_Novel-2H-isoquinolin-3-ones-as-antiplasmodial-falcipain-2-inhibitors_2009.pdf 484.5 KB
- 13/Shinonaga_Synthesis-and-structure-activity-relationships-of-radicicol-derivatives-and-WNT-5A-expression-inhibitory-activity_2009.pdf 484.2 KB
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- 17/Pacifico_Antioxidant-efficacy-of-iridoid-and-phenylethanoid-glycosides-from-the-medicinal-plant-Teucrium-chamaedris-in-cell-free-systems_2009.pdf 483.8 KB
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- 17/LaBeaume_Synthesis,-functionalization-and-photo-Bergman-chemistry-of-enediyne-bioconjugates_2009.pdf 476.9 KB
- 17/Leon_Tessaric-acid-derivatives-induce-G2M-cell-cycle-arrest-in-human-solid-tumor-cell-lines_2009.pdf 476.1 KB
- 24/8234-8240.pdf 475.3 KB
- 1/2009_17/01/0133.pdf 475.1 KB
- 18/Hu_Synthesis-and-activity-of-azaterphenyl-diamidines-against-Trypanosoma-brucei-rhodesiense-and-Plasmodium-falciparum_2009.pdf 473.8 KB
- 22/7816-7822.pdf 473.6 KB
- 14/Cressier_Synthesis,-antioxidant-properties-and-radioprotective-effects-of-new-benzothiazoles-and-thiadiazoles_2009.pdf 473.4 KB
- 3/sdarticle52.PDF 473.3 KB
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- 15/Nagy_Glucose-based-spiro-heterocycles-as-potent-inhibitors-of-glycogen-phosphorylase_2009.pdf 472.6 KB
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- 16/Marinec_Synthesis-of-orthogonally-reactive-FK506-derivatives-via-olefin-cross-metathesis_2009.pdf 467.8 KB
- 15/Loaiza_Parallel-synthesis-of-potent-dopaminergic-N-phenyltriazole-carboxamides-applying-a-novel-click-chemistry-based-phenol-linker_2009.pdf 467.5 KB
- 13/Asano_Synthesis-and-structure-activity-relationships-of-N-(4-amino-2,6-diisopropylphenyl)-N'-(1,4-diarylpiperidine-4-yl)methylureas-as-anti-hyperlipidemic-agents_2009.pdf 466.3 KB
- 14/Eissa_Synthesis,-biological-evaluation-and-docking-studies-of-novel-benzopyranone-congeners-for-their-expected-activity-as-anti-inflammatory,-analgesic-and-antipyretic-agents_2009.pdf 465.4 KB
- 7/sdarticle15.PDF 463.4 KB
- 18/Pettit_E-Combretastatin-and-E-resveratrol-structural-modifications-Antimicrobial-and-cancer-cell-growth-inhibitory-[beta]-E-nitrostyrenes_2009.pdf 462.5 KB
- 18/Sheng_Design,-synthesis-and-evaluation-of-flavonoid-derivatives-as-potent-AChE-inhibitors_2009.pdf 462.4 KB
- 4/sdarticle40.PDF 462.3 KB
- 18/Andersson_[omega]-Conotoxin-GVIA-mimetics-based-on-an-anthranilamide-core-Effect-of-variation-in-ammonium-side-chain-lengths-and-incorporation-of-fluorine_2009.pdf 462.2 KB
- 18/Ohtsuki_Death-receptor-5-promoter-enhancing-compounds-isolated-from-Catimbium-speciosum-and-their-enhancement-effect-on-TRAIL-induced-apoptosis_2009.pdf 460.2 KB
- 21/7606_7614.pdf 459.6 KB
- 17/Suzuki_Preparation-of-conophylline-affinity-nano-beads-and-identification-of-a-target-protein_2009.pdf 459.0 KB
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- 18/Tseng_Furo[3',2'3,4]naphtho[1,2-d]imidazole-derivatives-as-potential-inhibitors-of-inflammatory-factors-in-sepsis_2009.pdf 458.0 KB
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- 18/Wnuk_Inhibition-of-S-ribosylhomocysteinase-(LuxS)-by-substrate-analogues-modified-at-the-ribosyl-C-3-position_2009.pdf 454.6 KB
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- 13/Ishiyama_Synthesis-of-hybrid-analogues-of-caffeine-and-eudistomin-D-and-its-affinity-for-adenosine-receptors_2009.pdf 450.6 KB
- 5/sdarticle38.PDF 450.5 KB
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- 1/2009_17/01/0141.pdf 448.9 KB
- 13/Homma_Novel-hyaluronic-acid-methotrexate-conjugates-for-osteoarthritis-treatment_2009.pdf 447.8 KB
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- 13/Markl_Synthesis-and-pharmacological-evaluation-of-1,2,3,4-tetrahydropyrazino[1,2-a]indole-and-2-[(phenylmethylamino)methyl]-1H-indole-analogues-as-novel-melatoninergic-ligands_2009.pdf 445.6 KB
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- 14/Wang_Synthesis-of-amyloid-[beta]-peptide-1-42-(E22[Delta])-click-peptide-pH-triggered-in-situ-production-of-its-native-form_2009.pdf 442.2 KB
- 2/sdarticle10.PDF 441.9 KB
- 16/Matsuda_Melanogenesis-inhibitors-from-the-rhizomes-of-Alpinia-officinarum-in-B16-melanoma-cells_2009.pdf 441.8 KB
- 14/Zhang_`Click'-D1-receptor-agonists-with-a-5-HT1A-receptor-pharmacophore-producing-D2-receptor-activity_2009.pdf 441.8 KB
- 14/Bernotas_Novel-1-aminoethyl-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines-are-potent-5-HT6-agonists_2009.pdf 441.7 KB
- 20/7281-7289.pdf 441.6 KB
- 24/Graphical contents list.pdf 440.1 KB
- 14/Shah_In-vitro-erythrocytic-uptake-studies-of-artemisinin-and-selected-derivatives-using-LC-MS-and-2D-QSAR-analysis-of-uptake-in-parasitized-erythrocytes_2009.pdf 439.6 KB
- 20/7313-7323.pdf 437.8 KB
- 18/Paula_Design,-synthesis,-and-biological-evaluation-of-hydroquinone-derivatives-as-novel-inhibitors-of-the-sarcoendoplasmic-reticulum-calcium-ATPase_2009.pdf 436.6 KB
- 22/7647-7657.pdf 435.6 KB
- 14/Sugao_NF[kappa]B-decoy-delivery-using-dendritic-poly(l-lysine)-for-treatment-of-endotoxin-induced-hepatitis-in-mice_2009.pdf 434.8 KB
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- 14/Paulsen_In-vitro-biological-activity-and-structural-analysis-of-2,4-diamino-5-(2'-arylpropargyl)pyrimidine-inhibitors-of-Candida-albicans_2009.pdf 433.8 KB
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- 15/Petrelli_Selective-inhibition-of-nicotinamide-adenine-dinucleotide-kinases-by-dinucleoside-disulfide-mimics-of-nicotinamide-adenine-dinucleotide-analogues_2009.pdf 432.0 KB
- 11/sdarticle32.PDF 431.6 KB
- 15/Santos_Synthesis,-antiviral-activity-and-molecular-modeling-of-oxoquinoline-derivatives_2009.pdf 431.4 KB
- 4/sdarticle19.PDF 429.5 KB
- 24/8143-8148.pdf 429.3 KB
- 3/sdarticle53.PDF 428.5 KB
- 17/Sunduru_Synthesis-of-oxalamide-and-triazine-derivatives-as-a-novel-class-of-hybrid-4-aminoquinoline-with-potent-antiplasmodial-activity_2009.pdf 427.6 KB
- 12/4047-4063.pdf 427.5 KB
- 13/Nakamura_Discovery-of-tetrahydrotetramethylnaphthalene-analogs-as-adult-T-cell-leukemia-cell-selective-proliferation-inhibitors-in-a-small-chemical-library-constructed-based-on-multi-templ.pdf 425.2 KB
- 2/sdarticle47.PDF 424.0 KB
- 13/Saito_Synthesis-of-2[alpha]-propoxy-1[alpha],25-dihydroxyvitamin-D3-and-comparison-of-its-metabolism-by-human-CYP24A1-and-rat-CYP24A1_2009.pdf 423.5 KB
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- 14/Celen_Synthesis-and-biological-evaluation-of-11C-labeled-[beta]-galactosyl-triazoles-as-potential-PET-tracers-for-in-vivo-LacZ-reporter-gene-imaging_2009.pdf 417.6 KB
- 1/2009_17/01/0195.pdf 417.5 KB
- 14/Pudziuvelyte_Synthesis-and-antiproliferative-activity-of-2,4-disubstituted-6-aryl-7H-pyrrolo[3,2-d]pyrimidin-7-one-5-oxides_2009.pdf 417.0 KB
- 17/Liu_Synthesis-and-biological-evaluation-of-3,4-diaryl-5-aminoisoxazole-derivatives_2009.pdf 416.4 KB
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- 13/Charupant_Chemistry-of-renieramycins.-Part-8-Synthesis-and-cytotoxicity-evaluation-of-renieramycin-M-jorunnamycin-A-analogues_2009.pdf 414.2 KB
- 13/Pu_Synthesis-and-structure-activity-relationship-of-a-novel-series-of-heterocyclic-sulfonamide-[gamma]-secretase-inhibitors_2009.pdf 413.3 KB
- 8/sdarticle21.PDF 413.2 KB
- 20/7131-7137.pdf 412.0 KB
- 14/Gunosewoyo_Purinergic-P2X7-receptor-antagonists-Chemistry-and-fundamentals-of-biological-screening_2009.pdf 411.5 KB
- 21/7500_7509.pdf 410.9 KB
- 16/Zhan_Synthesis-and-biological-evaluation-of-imidazole-thioacetanilides-as-novel-non-nucleoside-HIV-1-reverse-transcriptase-inhibitors_2009.pdf 410.5 KB
- 13/Hasinoff_The-structure-based-design,-synthesis,-and-biological-evaluation-of-DNA-binding-amide-linked-bisintercalating-bisanthrapyrazole-anticancer-compounds_2009.pdf 410.5 KB
- 23/8086.pdf 410.4 KB
- 19/6908_6913.pdf 410.0 KB
- 14/Abdellatif_Diazen-1-ium-1,2-diolated-nitric-oxide-donor-ester-prodrugs-of-5-(4-carboxymethylphenyl)-1-(4-methanesulfonylphenyl)-3-trifluoromethyl-1H-pyrazole-and-its-aminosulfonyl-analog-S.pdf 409.7 KB
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- 6/sdarticle19.PDF 408.9 KB
- 23/8048.pdf 407.3 KB
- 16/Ribic_Novel-mannosyl-derivatives-of-peptidoglycan-monomer-Synthesis-and-biological-evaluation-of-immunomodulatory-properties_2009.pdf 406.6 KB
- 6/sdarticle36.PDF 405.9 KB
- 2/sdarticle8.PDF 405.8 KB
- 13/Ng_Potential-antioxidants-and-tyrosinase-inhibitors-from-synthetic-polyphenolic-deoxybenzoins_2009.pdf 405.2 KB
- 1/2009_17/01/0049.pdf 404.9 KB
- 6/sdarticle59.PDF 404.6 KB
- 14/Tanaka_Novel-3[alpha]-methoxyserrat-14-en-21[beta]-ol-(PJ-1)-and-3[beta]-methoxyserrat-14-en-21[beta]-ol-(PJ-2)-curcumin,-kojic-acid,-quercetin,-and-baicalein-conjugates-as-HIV-agents_2009.pdf 404.6 KB
- 22/7670-7679.pdf 404.1 KB
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- 10/sdarticle3.PDF 401.9 KB
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- 21/7585_7592.pdf 399.5 KB
- 6/sdarticle40.PDF 398.3 KB
- 3/sdarticle31.PDF 398.0 KB
- 14/Vardanyan_Synthesis-and-investigations-of-double-pharmacophore-ligands-for-treatment-of-chronic-and-neuropathic-pain_2009.pdf 397.4 KB
- 24/8149-8160.pdf 396.9 KB
- 11/sdarticle26.PDF 396.4 KB
- 14/Sauer_Synthesis-of-uracil-nucleotide-analogs-with-a-modified,-acyclic-ribose-moiety-as-P2Y2-receptor-antagonists_2009.pdf 396.2 KB
- 13/Innocenti_Carbonic-anhydrase-inhibitors.-Inhibition-and-homology-modeling-studies-of-the-fungal-[beta]-carbonic-anhydrase-from-Candida-albicans-with-sulfonamides_2009.pdf 396.1 KB
- 10/sdarticle8.PDF 394.9 KB
- 15/Bernini_A-novel-and-efficient-synthesis-of-highly-oxidized-lignans-by-a-methyltrioxorheniumhydrogen-peroxide-catalytic-system.-Studies-on-their-apoptogenic-and-antioxidant-activity_2009.pdf 394.9 KB
- 10/sdarticle19.PDF 394.0 KB
- 22/7723-7731.pdf 393.1 KB
- 11/sdarticle21.PDF 391.6 KB
- 18/Iwaniuk_Synthesis-and-antimalarial-activity-of-new-chloroquine-analogues-carrying-a-multifunctional-linear-side-chain_2009.pdf 391.3 KB
- 17/Cagnoni_Synthesis-of-pentopyranosyl-containing-thiodisaccharides.-Inhibitory-activity-against-[beta]-glycosidases_2009.pdf 391.0 KB
- 17/Gouy_Special-feature-of-mixed-phosphotriester-derivatives-of-cytarabine_2009.pdf 390.4 KB
- 19/6993_7001.pdf 390.4 KB
- 3/sdarticle40.PDF 390.0 KB
- 6/sdarticle7.PDF 388.5 KB
- 15/Liu_Synthesis-and-evaluation-of-a-novel-series-of-quinoline-derivatives-with-immunosuppressive-activity_2009.pdf 388.0 KB
- 21/7449_7456.pdf 387.1 KB
- 20/7138-7144.pdf 386.9 KB
- 23/7915.pdf 386.2 KB
- 4/sdarticle6.PDF 386.1 KB
- 21/7542_7547.pdf 385.8 KB
- 19/6942_6951.pdf 385.7 KB
- 15/Castagnolo_Synthesis,-biological-evaluation,-and-SAR-study-of-novel-pyrazole-analogues-as-inhibitors-of-Mycobacterium-tuberculosis-Part-2.-Synthesis-of-rigid-pyrazolones_2009.pdf 385.2 KB
- 3/sdarticle55.PDF 384.7 KB
- 11/sdarticle3.PDF 384.1 KB
- 11/sdarticle18.PDF 383.6 KB
- 17/Onnis_Synthesis-and-evaluation-of-anticancer-activity-of-2-arylamino-6-trifluoromethyl-3-(hydrazonocarbonyl)pyridines_2009.pdf 383.6 KB
- 9/sdarticle9.PDF 383.4 KB
- 13/Zhu_Synthesis-and-biological-evaluation-of-febrifugine-analogues-as-potential-antimalarial-agents_2009.pdf 383.4 KB
- 9/sdarticle23.PDF 381.5 KB
- 21/7510_7516.pdf 381.2 KB
- 13/Linz_Design,-synthesis-and-dopamine-D4-receptor-binding-activities-of-new-N-heteroaromatic-56-ring-Mannich-bases_2009.pdf 381.0 KB
- 4/sdarticle30.PDF 381.0 KB
- 15/Coi_Predictive-models,-based-on-classification-algorithms,-for-compounds-potentially-active-as-mitochondrial-ATP-sensitive-potassium-channel-openers_2009.pdf 380.7 KB
- 8/sdarticle4.PDF 380.2 KB
- 3/sdarticle33.PDF 379.8 KB
- 7/sdarticle10.PDF 379.3 KB
- 19/6890_6897.pdf 379.1 KB
- 1/2009_17/01/0119.pdf 376.8 KB
- 13/Lee_p-Terphenyls-from-the-fruiting-bodies-of-Paxillus-curtisii-and-their-antioxidant-properties_2009.pdf 376.7 KB
- 2/sdarticle40.PDF 374.3 KB
- 20/7248-7253.pdf 373.1 KB
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- 8/sdarticle9.PDF 372.0 KB
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- 19/7052_7055.pdf 371.2 KB
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- 16/Macone_Chromane-derivatives-of-small-aromatic-molecules-Chemoenzymatic-synthesis-and-growth-inhibitory-activity-on-human-tumor-cell-line-LoVo-WT_2009.pdf 371.1 KB
- 3/sdarticle8.PDF 370.7 KB
- 3/sdarticle21.PDF 369.7 KB
- 22/7775-7782.pdf 369.4 KB
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- 1/2009_17/01/0385.pdf 367.6 KB
- 3/sdarticle30.PDF 367.5 KB
- 18/Wecksler_Substrate-specificity-effects-of-lipoxygenase-products-and-inhibitors-on-soybean-lipoxygenase-1_2009.pdf 367.5 KB
- 18/Odagami_Identification-of-new-agonists-of-urotensin-II-from-a-cyclic-peptide-library_2009.pdf 366.8 KB
- 5/sdarticle29.PDF 365.4 KB
- 3/sdarticle28.PDF 365.3 KB
- 21/7429_7434.pdf 365.1 KB
- 17/Gnaccarini_Fluorometric-assay-for-tissue-transglutaminase-mediated-transamidation-activity_2009.pdf 364.4 KB
- 2/sdarticle22.PDF 364.3 KB
- 1/2009_17/01/0242.pdf 364.1 KB
- 4/sdarticle17.PDF 364.0 KB
- 14/Jin_Synthesis-and-structure-activity-relationship-of-3[beta]-(4-alkylthio,--methylsulfinyl,-and--methylsulfonylphenyl)tropane-and-3[beta]-(4-alkylthiophenyl)nortropane-derivatives-for-mono.pdf 363.7 KB
- 13/Paulino_Evaluation-of-anti-inflammatory-effect-of-synthetic-1,5-bis(4-acetoxy-3-methoxyphenyl)-1,4-pentadien-3-one,-HB2_2009.pdf 363.0 KB
- 14/Xu_Toward-preparation-of-antibody-based-imaging-probe-libraries-for-dual-modality-positron-emission-tomography-and-fluorescence-imaging_2009.pdf 362.0 KB
- 14/Kobayashi_A-new-small-molecule-that-directly-inhibits-the-DNA-binding-of-NF-[kappa]B_2009.pdf 361.5 KB
- 4/sdarticle12.PDF 361.4 KB
- 7/sdarticle29.PDF 361.0 KB
- 1/2009_17/01/0368.pdf 360.5 KB
- 8/sdarticle17.PDF 360.2 KB
- 8/sdarticle27.PDF 359.7 KB
- 6/sdarticle26.PDF 358.9 KB
- 23/7949.pdf 358.1 KB
- 20/7227-7238.pdf 357.6 KB
- 3/sdarticle57.PDF 357.3 KB
- 17/Zhan_1,2,3-Selenadiazole-thioacetanilides-Synthesis-and-anti-HIV-activity-evaluation_2009.pdf 356.6 KB
- 21/7562_7571.pdf 355.7 KB
- 11/sdarticle9.PDF 355.5 KB
- 15/Calderone_NO-glibenclamide-derivatives-Prototypes-of-a-new-class-of-nitric-oxide-releasing-anti-diabetic-drugs_2009.pdf 355.3 KB
- 21/7435_7440.pdf 355.1 KB
- 4/sdarticle42.PDF 354.4 KB
- 17/Chang_Microbial-transformation-of-isosteviol-oxime-and-the-inhibitory-effects-on-NF-[kappa]B-and-AP-1-activation-in-LPS-stimulated-macrophages_2009.pdf 353.4 KB
- 5/sdarticle11.PDF 352.4 KB
- 14/Tevyashova_Reaction-of-the-antitumor-antibiotic-olivomycin-I-with-aryl-diazonium-salts.-Synthesis,-cytotoxic-and-antiretroviral-potency-of-5-aryldiazenyl-6-O-deglycosyl-derivatives-of-oliv.pdf 352.1 KB
- 20/7362-7367.pdf 351.4 KB
- 19/6872_6878.pdf 350.2 KB
- 15/Sadler_Synthetic-strategies-toward-carbocyclic-purine-pyrimidine-hybrid-nucleosides_2009.pdf 349.3 KB
- 2/sdarticle37.PDF 349.1 KB
- 20/7275-7280.pdf 348.1 KB
- 6/sdarticle30.PDF 348.0 KB
- 6/sdarticle10.PDF 348.0 KB
- 13/Lee_Quinazolindione-derivatives-as-potent-5-HT3A-receptor-antagonists_2009.pdf 345.6 KB
- 14/Zarghi_Synthesis-and-biological-evaluation-of-new-4-carboxyl-quinoline-derivatives-as-cyclooxygenase-2-inhibitors_2009.pdf 345.4 KB
- 15/Langkjaer_UNA-(unlocked-nucleic-acid)-A-flexible-RNA-mimic-that-allows-engineering-of-nucleic-acid-duplex-stability_2009.pdf 344.9 KB
- 18/Czako_Synthesis-and-glycogen-phosphorylase-inhibitory-activity-of-N-([beta]-d-glucopyranosyl)amides-possessing-1,4-benzodioxane-moiety_2009.pdf 343.9 KB
- 9/sdarticle8.PDF 343.6 KB
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- 19/7015_7020.pdf 342.2 KB
- 13/Herm_N-Substituted-2-alkyl--and-2-arylnorapomorphines-Novel,-highly-active-D2-agonists_2009.pdf 341.2 KB
- 19/7008_7014.pdf 340.8 KB
- 1/2009_17/01/0189.pdf 340.3 KB
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- 2/sdarticle19.PDF 334.0 KB
- 16/Suzuki_Design,-synthesis,-enzyme-inhibition,-and-tumor-cell-growth-inhibition-of-2-anilinobenzamide-derivatives-as-SIRT1-inhibitors_2009.pdf 332.6 KB
- 15/Kumar_Design-and-synthesis-of-an-all-in-one-3-(1,1-difluoroprop-2-ynyl)-3H-diazirin-3-yl-functional-group-for-photo-affinity-labeling_2009.pdf 332.2 KB
- 9/sdarticle26.PDF 331.7 KB
- 19/6796_6802.pdf 330.6 KB
- 7/sdarticle7.PDF 329.3 KB
- 17/Watanabe_Synthesis-and-biological-evaluation-of-radioiodinated-2,5-diphenyl-1,3,4-oxadiazoles-for-detecting-[beta]-amyloid-plaques-in-the-brain_2009.pdf 328.1 KB
- 7/sdarticle27.PDF 325.4 KB
- 13/Verhaeghe_Synthesis-and-in-vitro-antiplasmodial-evaluation-of-4-anilino-2-trichloromethylquinazolines_2009.pdf 325.0 KB
- 1/2009_17/01/0411.pdf 324.7 KB
- 8/sdarticle10.PDF 320.2 KB
- 1/2009_17/01/0303.pdf 319.5 KB
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- 20/7126-7130.pdf 316.8 KB
- 16/Dangate_2-O-[beta]-d-Glucopyranosyl-sn-glycerol-based-analogues-of-sulfoquinovosyldiacylglycerols-(SQDG)-and-their-role-in-inhibiting-Epstein-Barr-virus-early-antigen-activation_2009.pdf 316.5 KB
- 18/Zhuang_Synthesis-and-biological-evaluation-of-4-fluoroproline-and-4-fluoropyrrolidine-2-acetic-acid-derivatives-as-new-GABA-uptake-inhibitors_2009.pdf 315.3 KB
- 14/Ranga-Rao_New-furanoflavanoids,-intestinal-[alpha]-glucosidase-inhibitory-and-free-radical-(DPPH)-scavenging,-activity-from-antihyperglycemic-root-extract-of-Derris-indica-(Lam.)_2009.pdf 314.9 KB
- 17/Obando_Synthesis,-antifungal,-haemolytic-and-cytotoxic-activities-of-a-series-of-bis(alkylpyridinium)alkanes_2009.pdf 314.2 KB
- 11/sdarticle24.PDF 314.1 KB
- 14/Guzel_Carbonic-anhydrase-inhibitors.-Aromaticheterocyclic-sulfonamides-incorporating-phenacetyl,-pyridylacetyl-and-thienylacetyl-tails-act-as-potent-inhibitors-of-human-mitochondrial-isofo.pdf 314.1 KB
- 11/sdarticle33.PDF 312.5 KB
- 12/4096-4105.pdf 312.4 KB
- 6/sdarticle12.PDF 312.4 KB
- 15/Usera_`Novel-alkyl-side-chain-sulfone-1[alpha],25-dihydroxyvitamin-D3-analogs-A-comparison-of-in-vitro-antiproliferative-activities-and-in-vivo-calcemic-activities'_2009.pdf 312.0 KB
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- 18/Balo_Synthesis-and-pharmacological-evaluation-of-novel-1--and-8-substituted-3-furfuryl-xanthines-as-adenosine-receptor-antagonists_2009.pdf 309.2 KB
- 1/2009_17/01/0270.pdf 307.9 KB
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- 16/Konno_Synthesis-of-[19,-35,-36-13C3]-labeled-TAK779-as-a-molecular-probe_2009.pdf 306.0 KB
- 2/sdarticle38.PDF 304.1 KB
- 1/2009_17/01/0235.pdf 304.1 KB
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- 17/Beauchard_Synthesis-and-kinase-inhibitory-activity-of-novel-substituted-indigoids_2009.pdf 303.4 KB
- 22/7749-7754.pdf 302.3 KB
- 11/sdarticle8.PDF 302.1 KB
- 22/7630-7634.pdf 300.8 KB
- 15/Zarghi_Design-and-synthesis-of-new-1,3-benzthiazinan-4-one-derivatives-as-selective-cyclooxygenase-(COX-2)-inhibitors_2009.pdf 300.3 KB
- 1/2009_17/01/0337.pdf 298.9 KB
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- 1/2009_17/01/0418.pdf 295.4 KB
- 1/2009_17/01/0260.pdf 293.6 KB
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- 18/Ghirmai_Synthesis-and-pharmacological-evaluation-of-6-naltrexamine-analogs-for-alcohol-cessation_2009.pdf 292.4 KB
- 2/sdarticle4.PDF 292.3 KB
- 3/sdarticle38.PDF 291.4 KB
- 13/Tundis_Cytotoxic-activity-and-inhibitory-effect-on-nitric-oxide-production-of-triterpene-saponins-from-the-roots-of-Physospermum-verticillatum-(Waldst-&-Kit)-(Apiaceae)_2009.pdf 291.3 KB
- 14/Gibson_Enaminones-10.-Molecular-modeling-aspects-of-the-5-methylcyclohexenone-derivatives_2009.pdf 291.2 KB
- 3/sdarticle58.PDF 291.1 KB
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- 13/Jia_Synthesis-and-in-vitro-anti-hepatitis-B-virus-activity-of-6H-[1]benzothiopyrano[4,3-b]quinolin-9-ols_2009.pdf 290.5 KB
- 3/sdarticle46.PDF 289.0 KB
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- 1/2009_17/01/0222.pdf 288.2 KB
- 17/Yamashita_Synthesis-and-evaluation-of-bioactive-naphthoquinones-from-the-Brazilian-medicinal-plant,-Tabebuia-avellanedae_2009.pdf 288.2 KB
- 22/7823-7830.pdf 288.0 KB
- 16/Yamada_Synthesis-and-properties-of-nucleoside-derivatives-acylated-by-chemically-stable-2-(trimethylsilyl)benzoyl-group_2009.pdf 287.1 KB
- 4/sdarticle39.PDF 286.8 KB
- 6/sdarticle13.PDF 284.2 KB
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- 13/Mukai_Design-of-Ga-DOTA-based-bifunctional-radiopharmaceuticals-Two-functional-moieties-can-be-conjugated-to-radiogallium-DOTA-without-reducing-the-complex-stability_2009.pdf 282.4 KB
- 6/sdarticle15.PDF 282.4 KB
- 16/Turner_Structural-basis-for-[alpha]-conotoxin-potency-and-selectivity_2009.pdf 280.0 KB
- 4/sdarticle16.PDF 278.6 KB
- 13/Ioannou_9,11-Secosterols-with-antiproliferative-activity-from-the-gorgonian-Eunicella-cavolini_2009.pdf 277.2 KB
- 14/Donnici_Ruthenium-complexes-endowed-with-potent-anti-Trypanosoma-cruzi-activity-Synthesis,-biological-characterization-and-structure-activity-relationships_2009.pdf 277.0 KB
- 6/sdarticle16.PDF 276.7 KB
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- 18/Montes-Avila_Solution-phase-parallel-synthesis-of-substituted-chalcones-and-their-antiparasitary-activity-against-Giardia-lamblia_2009.pdf 272.7 KB
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- 17/Takano_Amphotericin-B-induced-ion-flux-is-markedly-attenuated-in-phosphatidylglycerol-membrane-as-evidenced-by-a-newly-devised-fluorometric-method_2009.pdf 266.4 KB
- 15/Nishimura_Discriminatory-synergistic-effect-of-Trp-substitutions-in-superagonist-[(ArgLys)14,-(ArgLys)15]nociceptin-on-ORL1-receptor-binding-and-activation_2009.pdf 266.3 KB
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- 15/Baldisserotto_N-Terminal-prolonged-vinyl-ester-based-peptides-as-selective-proteasome-[beta]1-subunit-inhibitors_2009.pdf 261.1 KB
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